{"created":"2023-05-15T15:01:59.808251+00:00","id":84089,"links":{},"metadata":{"_buckets":{"deposit":"cb867d78-b770-4ea1-ab80-02173c3f28b6"},"_deposit":{"created_by":1,"id":"84089","owners":[1],"pid":{"revision_id":0,"type":"depid","value":"84089"},"status":"published"},"_oai":{"id":"oai:repo.qst.go.jp:00084089","sets":["1"]},"author_link":["1042271","1042258","1042259","1042269","1042263","1042275","1042270","1042273","1042253","1042261","1042254","1042265","1042272","1042276","1042267","1042257","1042266","1042274","1042256","1042268","1042255","1042262","1042264","1042260"],"item_8_biblio_info_7":{"attribute_name":"書誌情報","attribute_value_mlt":[{"bibliographicIssueDates":{"bibliographicIssueDate":"2021-10","bibliographicIssueDateType":"Issued"},"bibliographicPageEnd":"1135","bibliographicPageStart":"1127","bibliographicVolumeNumber":"49","bibliographic_titles":[{"bibliographic_title":"European journal of nuclear medicine and molecular imaging"}]}]},"item_8_description_5":{"attribute_name":"抄録","attribute_value_mlt":[{"subitem_description":"Histamine H receptor antagonists and inverse agonists have been extensively developed to treat sleep-wake, neurocognitive, and allied disorders. However, potential adverse effects, including insomnia, hampered the clinical use of these drugs, possibly due to their persistent interaction with the target molecules. The purpose of the present study was to estimate the pharmacokinetics and pharmacodynamics of enerisant, a novel antagonist and inverse agonist for histamine H receptors.","subitem_description_type":"Abstract"}]},"item_8_relation_13":{"attribute_name":"PubMed番号","attribute_value_mlt":[{"subitem_relation_type_id":{"subitem_relation_type_id_text":"34651222","subitem_relation_type_select":"PMID"}}]},"item_8_relation_14":{"attribute_name":"DOI","attribute_value_mlt":[{"subitem_relation_type_id":{"subitem_relation_type_id_text":"10.1007/s00259-021-05571-1","subitem_relation_type_select":"DOI"}}]},"item_8_relation_17":{"attribute_name":"関連サイト","attribute_value_mlt":[{"subitem_relation_type_id":{"subitem_relation_type_id_text":"https://link.springer.com/article/10.1007/s00259-021-05571-1","subitem_relation_type_select":"URI"}}]},"item_8_source_id_9":{"attribute_name":"ISSN","attribute_value_mlt":[{"subitem_source_identifier":"1619-7070","subitem_source_identifier_type":"ISSN"}]},"item_access_right":{"attribute_name":"アクセス権","attribute_value_mlt":[{"subitem_access_right":"metadata only 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Tetsuya"}],"nameIdentifiers":[{"nameIdentifier":"1042265","nameIdentifierScheme":"WEKO"}]},{"creatorNames":[{"creatorName":"Yasuyuki, Kimura","creatorNameLang":"en"}],"nameIdentifiers":[{"nameIdentifier":"1042266","nameIdentifierScheme":"WEKO"}]},{"creatorNames":[{"creatorName":"Keisuke, Takahata","creatorNameLang":"en"}],"nameIdentifiers":[{"nameIdentifier":"1042267","nameIdentifierScheme":"WEKO"}]},{"creatorNames":[{"creatorName":"Soichiro, Kitamura","creatorNameLang":"en"}],"nameIdentifiers":[{"nameIdentifier":"1042268","nameIdentifierScheme":"WEKO"}]},{"creatorNames":[{"creatorName":"Chie, Seki","creatorNameLang":"en"}],"nameIdentifiers":[{"nameIdentifier":"1042269","nameIdentifierScheme":"WEKO"}]},{"creatorNames":[{"creatorName":"Yoko, Ikoma","creatorNameLang":"en"}],"nameIdentifiers":[{"nameIdentifier":"1042270","nameIdentifierScheme":"WEKO"}]},{"creatorNames":[{"creatorName":"Masanori, 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[11C]TASP457."}]},"item_type_id":"8","owner":"1","path":["1"],"pubdate":{"attribute_name":"公開日","attribute_value":"2021-10-18"},"publish_date":"2021-10-18","publish_status":"0","recid":"84089","relation_version_is_last":true,"title":["Pharmacokinetic and pharmacodynamic assessment of histamine H3 receptor occupancy by enerisant: a human PET study with a novel H3 binding ligand, [11C]TASP457."],"weko_creator_id":"1","weko_shared_id":-1},"updated":"2023-05-15T17:21:56.542332+00:00"}