{"created":"2023-05-15T14:57:34.151296+00:00","id":78131,"links":{},"metadata":{"_buckets":{"deposit":"7511163d-6b1e-45e2-996c-6939ece163cd"},"_deposit":{"created_by":1,"id":"78131","owners":[1],"pid":{"revision_id":0,"type":"depid","value":"78131"},"status":"published"},"_oai":{"id":"oai:repo.qst.go.jp:00078131","sets":["1"]},"author_link":["1002109","1002115","1002107","1002121","1002116","1002110","1002108","1002112","1002104","1002103","1002124","1002106","1002123","1002102","1002111","1002117","1002120","1002122","1002114","1002105","1002118","1002101","1002119","1002113"],"item_8_biblio_info_7":{"attribute_name":"書誌情報","attribute_value_mlt":[{"bibliographicIssueDates":{"bibliographicIssueDate":"2019-12","bibliographicIssueDateType":"Issued"},"bibliographicIssueNumber":"4","bibliographicPageStart":"126879","bibliographicVolumeNumber":"30","bibliographic_titles":[{"bibliographic_title":"Bioorganic & Medicinal Chemistry Letters"}]}]},"item_8_description_5":{"attribute_name":"抄録","attribute_value_mlt":[{"subitem_description":"Transmembrane AMPA receptor regulatory proteins (TARPs) are a recently discovered family of proteins that modulate AMPA receptors activity. Based on a potent and selective TARP subtype γ-8 antagonist, 6-(methyl(4-(pyridin-2-yl)thiazol-2-yl)amino)benzo[d]thiazol-2(3H)-one (compound 9), we perform the radiosynthesis of its 11C-isotopologue 1 and conduct preliminary PET evaluation to test the feasibility of imaging TARP γ-8 dependent receptors in 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