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[(11)C]TASP457, a novel PET ligand for histamine H3 receptors in human brain.
https://repo.qst.go.jp/records/47492
https://repo.qst.go.jp/records/4749211695111-ef76-468d-b71d-3738f75ff12c
Item type | 学術雑誌論文 / Journal Article(1) | |||||
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公開日 | 2016-08-23 | |||||
タイトル | ||||||
タイトル | [(11)C]TASP457, a novel PET ligand for histamine H3 receptors in human brain. | |||||
言語 | ||||||
言語 | eng | |||||
資源タイプ | ||||||
資源タイプ識別子 | http://purl.org/coar/resource_type/c_6501 | |||||
資源タイプ | journal article | |||||
アクセス権 | ||||||
アクセス権 | metadata only access | |||||
アクセス権URI | http://purl.org/coar/access_right/c_14cb | |||||
著者 |
Kimura, Yasuyuki
× Kimura, Yasuyuki× Seki, Chie× Ikoma, Yoko× Ichise, Masanori× Kawamura, Kazunori× Takahata, Keisuke× Moriguchi, Sho× Nagashima, Tomohisa× Ishii, Tatsuya× Kitamura, Soichiro× Niwa, Fumitoshi× Endo, Hironobu× Yamada, Makiko× Higuchi, Makoto× Zhang, Ming-Rong× Suhara, Tetsuya× 木村 泰之× 関 千江× 生駒 洋子× 市瀬 正則× 河村 和紀× 高畑 圭輔× 森口 翔× 永嶌 朋久× 石井 辰弥× 北村 聡一郎× 丹羽 文俊× 遠藤 浩信× 山田 真希子× 樋口 真人× 張 明栄× 須原 哲也 |
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抄録 | ||||||
内容記述タイプ | Abstract | |||||
内容記述 | The histamine H3 receptors are presynaptic neuroreceptors that inhibit the release of histamine and other neurotransmitters. The receptors are considered a drug target for sleep disorders and neuropsychiatric disorders with cognitive decline. We developed a novel PET ligand for the H3 receptors, [(11)C]TASP0410457 ([(11)C]TASP457), with high affinity, selectivity and favorable kinetic properties in the monkey, and evaluated its kinetics and radiation safety profile for quantifying the H3 receptors in human brain. | |||||
書誌情報 |
European journal of nuclear medicine and molecular imaging 巻 43, 号 9, p. 1653-1663, 発行日 2016-02 |
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出版者 | ||||||
出版者 | Springer | |||||
ISSN | ||||||
収録物識別子タイプ | ISSN | |||||
収録物識別子 | 1619-7070 | |||||
PubMed番号 | ||||||
識別子タイプ | PMID | |||||
関連識別子 | 26902370 | |||||
DOI | ||||||
識別子タイプ | DOI | |||||
関連識別子 | 10.1007/s00259-016-3332-6 |